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Iso- and Benzisothiazolinone Inhibitors of Monoacylglycerol Lipase: Exploring On-Target Activity Through Scaffold Decoration and In Situ Warhead Generation.

Authors: Rocca E, Bedini A, Scalvini L, Galvani F, Castelli R, Sarcone L, Recchia A, Fanini F, Tran A, Rivara S, Spadoni G, Piomelli D, Mor M
Journal: ChemMedChem
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Abstract